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Found 424 Enz. Inhib. hit(s) with Target = 'Capsid scaffolding protein'
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133948((S)-2-[(3aS,6S,6aR)-4-(6-Hydroxymethyl-benzothiazo...)
Affinity DataKi:  0.310nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133960((S)-2-((3aS,6S,6aR)-4-Cyclopropanecarbonyl-6-methy...)
Affinity DataKi:  2nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133962((3S,3aR,6aS)-4-({(2S)-1-[(5-Chloro-3-methyl-1-benz...)
Affinity DataKi:  2nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133951(2-{(3S,3aR,6aS)-4-[(S)-1-(4-Isopropyl-phenylcarbam...)
Affinity DataKi:  7.40nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133981((2S)-2-{[(3aS,6S,6aR)-4-(Cyclopropylcarbonyl)-6-me...)
Affinity DataKi:  9nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133989((S)-2-((3aS,6S,6aR)-4-Cyclopropanecarbonyl-6-methy...)
Affinity DataKi:  9nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133952((S)-2-((3aS,6S,6aR)-4-Benzothiazol-2-yl-6-methyl-5...)
Affinity DataKi:  10nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133969((S)-2-((3aS,6S,6aR)-4-Cyclopropanecarbonyl-6-methy...)
Affinity DataKi:  15nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133957((S)-2-[(3aS,6S,6aR)-6-Methyl-4-((2R,3S)-2-(S)-meth...)
Affinity DataKi:  16nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133980((2S)-2-{[(3aS,6S,6aR)-4-(Cyclopropylcarbonyl)-6-me...)
Affinity DataKi:  18nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50107904((3S,3aR,6aS)-1-Cyclopropanecarbonyl-4-[(S)-1-(5-di...)
Affinity DataKi:  20nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133950((S)-2-[(3aS,6S,6aR)-6-Methyl-5-oxo-4-(6-trifluorom...)
Affinity DataKi:  20nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133992((3S,3aR,6aS)-4-[(S)-1-(Biphenyl-4-carbonyl)-pyrrol...)
Affinity DataKi:  21nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133953((S)-2-((3aS,6S,6aR)-6-Methyl-5-oxo-4-thiazolo[5,4-...)
Affinity DataKi:  21nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133975((S)-2-[(3aS,6S,6aR)-6-Methyl-4-(6-nitro-benzothiaz...)
Affinity DataKi:  25nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133978((3S,3aR,6aS)-1-Cyclopropanecarbonyl-3-methyl-4-[(S...)
Affinity DataKi:  33nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133964((3S,3aR,6aS)-1-Cyclopropanecarbonyl-3-methyl-4-[(S...)
Affinity DataKi:  33nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133977((2S)-2-{[(3aS,6S,6aR)-4-(Cyclopropylcarbonyl)-6-me...)
Affinity DataKi:  38nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133979((3S,3aR,6aS)-1-Cyclopropanecarbonyl-4-[(S)-1-(4-is...)
Affinity DataKi:  39nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133988((3S,3aR,6aS)-1-(Cyclopropylcarbonyl)-3-methyl-4-{[...)
Affinity DataKi:  40nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133985((S)-2-[(3aS,6S,6aR)-4-(6-Methoxy-benzothiazol-2-yl...)
Affinity DataKi:  43nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133949((3S,3aR,6aS)-1-Cyclopropanecarbonyl-3-methyl-4-[(S...)
Affinity DataKi:  60nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133991((3S,3aR,6aS)-1-Cyclopropanecarbonyl-3-methyl-4-[(S...)
Affinity DataKi:  79nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133954((3S,3aR,6aS)-1-Cyclopropanecarbonyl-3-methyl-4-[(S...)
Affinity DataKi:  79nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59224(Pepstatin analog, 12)
Affinity DataKi:  96nM IC50:  360nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133987((3S,3aR,6aS)-1-Cyclopropanecarbonyl-4-[(S)-1-(4-is...)
Affinity DataKi:  99nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59223(Pepstatin analog, 11)
Affinity DataKi:  175nM IC50:  730nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59213(Pepstatin analog, 1)
Affinity DataKi:  220nM IC50:  350nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50133967((S)-2-((3aS,6S,6aR)-6-Methyl-5-oxo-4-thiazol-2-yl-...)
Affinity DataKi:  446nMAssay Description:Potency against human cytomegalovirus protease in HCMV pNA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59220(Pepstatin analog, 8)
Affinity DataKi:  600nM IC50:  2.90E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59222(Pepstatin analog, 10)
Affinity DataKi:  650nM IC50:  2.50E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59219(Pepstatin analog, 7)
Affinity DataKi:  720nM IC50:  2.70E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59216(Pepstatin analog, 4)
Affinity DataKi:  1.13E+3nM IC50:  4.40E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59217(Pepstatin analog, 5)
Affinity DataKi:  1.29E+3nM IC50:  4.90E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University

LigandPNGBDBM59214(Pepstatin analog, 2)
Affinity DataKi:  3.00E+3nM IC50:  5.90E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143640(4-({5-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-napht...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143634(4-{[5-(4-Bromo-phenoxymethyl)-naphthalen-2-ylamino...)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143650(4-{[5-(3-Chloro-phenoxymethyl)-naphthalen-2-ylamin...)
Affinity DataIC50:  3.10nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143617(CHEMBL442168 | N-{5-[2-(8-Chloro-quinolin-2-yl)-vi...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143630(CHEMBL299043 | N-{5-[(E)-2-(6-Chloro-quinolin-2-yl...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143627(C,C,C-Trifluoro-N-{5-[2-(6-methoxy-quinolin-2-yl)-...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143623(CHEMBL299278 | N-{5-[2-(6-Dimethylamino-quinolin-2...)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143637(CHEMBL56633 | N-{5-[2-(4-Chloro-phenyl)-vinyl]-nap...)
Affinity DataIC50:  4.30nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143633(4-chloro-N-[({5-[(1E)-7-chloroquinolin-2-yl)vinyl]...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143616(4-[(5-Phenoxymethyl-naphthalen-2-ylamino)-methyl]-...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143621(CHEMBL55390 | N-[5-(3-Chloro-benzyloxy)-naphthalen...)
Affinity DataIC50:  5.10nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143638(CHEMBL57565 | N-[5-(3-Bromo-benzyloxy)-naphthalen-...)
Affinity DataIC50:  6.10nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143628(C,C,C-Trifluoro-N-{5-[2-(6-methyl-quinolin-2-yl)-v...)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143641(C,C,C-Trifluoro-N-{5-[2-(3-trifluoromethyl-phenyl)...)
Affinity DataIC50:  6.5nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143618(C,C,C-Trifluoro-N-{5-[2-(3-methoxy-phenyl)-vinyl]-...)
Affinity DataIC50:  6.60nMAssay Description:Inhibitory concentration against HCMV protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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