Compile Data Set for Download or QSAR
maximum 50k data
Found 174 Enz. Inhib. hit(s) with Target = 'Isoleucine--tRNA ligase'
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524451(CHEMBL4553017)
Affinity DataKi:  1.20nMAssay Description:Inhibition of recombinant Escherichia coli BL21(DE3) isoleucyl-tRNA synthetase expressed in Escherichia coli Rosetta 2 (DE3) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50222902(CHEMBL1163069)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50290686(9-((E)-4-((2S,3R,4R,5S)-3,4-dihydroxy-5-(((2S,3S)-...)
Affinity DataKi:  2.5nMAssay Description:Competitive inhibition of Escherichia coli Isoleucyl-tRNA synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524360(CHEMBL3265242)
Affinity DataKi:  17nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524354(CHEMBL3265243)
Affinity DataKi:  55nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544145(CHEMBL4636583)
Affinity DataKi:  88nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544146(CHEMBL4648043)
Affinity DataKi:  114nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458120(CHEMBL4215986)
Affinity DataKi:  213nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524358(CHEMBL4475568)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18152((2S,3S)-2-amino-3,4-dimethylpentanoic acid | L-2-A...)
Affinity DataKi:  4.55E+4nM ΔG°:  -24.4kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18150((2S,3S)-2-amino-3-methylhexanoic acid | L-2-Amino-...)
Affinity DataKi:  5.00E+4nM ΔG°:  -24.1kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18149((3S)-2-amino-3-methylhexanoic acid | DL-2-Amino-3S...)
Affinity DataKi:  5.88E+4nM ΔG°:  -23.7kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18144(2-amino-3-ethylpentanoic acid | DL-2-Amino-3-ethyl...)
Affinity DataKi:  5.30E+5nM ΔG°:  -18.4kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18145((2S)-2-amino-3-ethylpentanoic acid | L-2-Amino-3-e...)
Affinity DataKi:  5.60E+5nM ΔG°:  -18.2kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18146(2-amino-3,3-dimethylpentanoic acid | DL-2-Amino-3,...)
Affinity DataKi:  1.25E+6nM ΔG°:  -16.3kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18151((3R)-2-amino-3-methylhexanoic acid | DL-2-Amino-3R...)
Affinity DataKi:  1.67E+6nM ΔG°:  -15.6kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18141((2S,4S)-2-amino-4-methylhexanoic acid | L-2-Amino-...)
Affinity DataKi:  2.00E+6nM ΔG°:  -15.1kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18155((3S)-2-amino-3-methylheptanoic acid | DL-2-Amino-3...)
Affinity DataKi:  2.50E+6nM ΔG°:  -14.6kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18143((2S)-2-amino-5-methylhexanoic acid | L-2-Amino-5-m...)
Affinity DataKi:  2.50E+6nM ΔG°:  -14.6kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18153((3R)-2-amino-3,4-dimethylpentanoic acid | DL-2-Ami...)
Affinity DataKi:  3.33E+6nM ΔG°:  -13.9kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18142(2-amino-5-methylhexanoic acid | DL-2-Amino-5-methy...)
Affinity DataKi:  3.33E+6nM ΔG°:  -13.9kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18154((2S,3R)-2-amino-3,4-dimethylpentanoic acid | L-2-A...)
Affinity DataKi:  5.00E+6nM ΔG°:  -12.9kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18158((3R)-2-amino-3-ethylhexanoic acid | DL-2-Amino-3R-...)
Affinity DataKi:  5.00E+6nM ΔG°:  -12.9kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18157((3S)-2-amino-3-ethylhexanoic acid | DL-2-Amino-3S-...)
Affinity DataKi:  5.00E+6nM ΔG°:  -12.9kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18159((2S)-2-amino-3-methylpentan-1-ol | L-isoleucinol)
Affinity DataKi:  8.33E+6nM ΔG°:  -11.7kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18148((2S)-2-amino-4,4-dimethylpentanoic acid | L-2-Amin...)
Affinity DataKi:  1.25E+7nM ΔG°:  -10.7kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18147(2-amino-4,4-dimethylpentanoic acid | DL-2-Amino-4,...)
Affinity DataKi:  1.25E+7nM ΔG°:  -10.7kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18160((2S)-2-amino-3-methylbutan-1-ol | L-Valinol)
Affinity DataKi:  1.43E+7nM ΔG°:  -10.4kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18139((2S)-2-aminoheptanoic acid | L-2-Amino-heptanoic a...)
Affinity DataKi:  1.67E+7nM ΔG°:  -9.98kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM18156((3R)-2-amino-3-methylheptanoic acid | DL-2-Amino-3...)
Affinity DataKi:  1.67E+7nM ΔG°:  -9.98kJ/molepH: 7.5 T: 2°CAssay Description:Utilizing an analytical ultracentrifuge, the binding constants of various amino acids and isoleucine analogues to IleRS were estimated from their com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471296(CHEMBL87935)
Affinity DataIC50:  0.700nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290686(9-((E)-4-((2S,3R,4R,5S)-3,4-dihydroxy-5-(((2S,3S)-...)
Affinity DataIC50:  0.800nMAssay Description:Compound was evaluated for inhibitory activity against Isoleucyl-tRNA synthetaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50290686(9-((E)-4-((2S,3R,4R,5S)-3,4-dihydroxy-5-(((2S,3S)-...)
Affinity DataIC50:  0.850nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471292(CHEMBL315230)
Affinity DataIC50:  1.10nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471294(CHEMBL276855)
Affinity DataIC50:  1.90nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471297(CHEMBL424608)
Affinity DataIC50:  2.10nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471293(CHEMBL83449)
Affinity DataIC50:  3.60nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470911(CHEMBL122825)
Affinity DataIC50:  4.45nMAssay Description:Inhibitory activity against isoleucyl-tRNA synthetase (IRS) of Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50217841(REVEROMYCIN A)
Affinity DataIC50:  4.46nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471295(CHEMBL312853)
Affinity DataIC50:  5.30nMAssay Description:Inhibition concentration against Isoleucyl-tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50471291(CHEMBL83394)
Affinity DataIC50:  6nMAssay Description:Inhibition concentration against isoleucyl tRNA synthetase from Staphylococcus aureus NCTC 6571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470914(CHEMBL120343)
Affinity DataIC50:  6.67nMAssay Description:Inhibitory activity against isoleucyl-tRNA synthetase (IRS) of Staphylococcus aureus NCTC 3571More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524451(CHEMBL4553017)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of recombinant Escherichia coli BL21(DE3) isoleucyl-tRNA synthetase expressed in Escherichia coli Rosetta 2 (DE3) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470913(CHEMBL120798)
Affinity DataIC50:  6.87nMAssay Description:Inhibitory activity against isoleucyl-tRNA synthetase (IRS) of Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470912(CHEMBL120437)
Affinity DataIC50:  7.98nMAssay Description:Inhibitory activity against isoleucyl-tRNA synthetase (IRS) of Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50093003((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)
Affinity DataIC50:  14nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366870(CHEMBL605376)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against Escherichia coli Isoleucyl-tRNA synthetase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Trypanosoma brucei (Kinetoplastids))
University Of Washington

LigandPNGBDBM188488(NSC70422)
Affinity DataIC50:  14.1nMAssay Description:Compound stocks were prepared at a 10 mM concentration in dimethyl sulfoxide.T. brucei bloodstream forms (100 µl at 2.0 × 10^4 parasites/ml) were pla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50075058(((S)-2-Amino-3-methyl-pentanoyl)-sulfamic acid (2R...)
Affinity DataIC50:  15nMAssay Description:Compound tested for the inhibition of human isoleucyl-tRNA synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50479281(2,3-DIHYDROREVEROMYCIN A)
Affinity DataIC50:  17.5nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 174 total ) | Next | Last >>
Jump to: