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Found 652 Enz. Inhib. hit(s) with Target = 'Kallikrein-7'
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50125021(CHEMBL3623779)
Affinity DataKi:  0.800nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Mus musculus)
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50598266(CHEMBL5203652)
Affinity DataKi:  4.10nMAssay Description:Inhibition of mouse KLK7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598311(CHEMBL5185665)
Affinity DataKi:  7nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598297(CHEMBL5198206)
Affinity DataKi:  8.80nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598292(CHEMBL5173572)
Affinity DataKi:  9nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598306(CHEMBL5173148)
Affinity DataKi:  10nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598296(CHEMBL5179139)
Affinity DataKi:  12nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598309(CHEMBL5204039)
Affinity DataKi:  16nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50124906(CHEMBL3623776)
Affinity DataKi:  17nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598301(CHEMBL5189873)
Affinity DataKi:  18nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598305(CHEMBL5191378)
Affinity DataKi:  19nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598310(CHEMBL5185516)
Affinity DataKi:  29nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598295(CHEMBL5175658)
Affinity DataKi:  29nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598288(CHEMBL5204199)
Affinity DataKi:  31nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598291(CHEMBL5177855)
Affinity DataKi:  32nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598307(CHEMBL5177530)
Affinity DataKi:  36nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113060(US9695194, 1)
Affinity DataKi:  48nM ΔG°:  -43.5kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598303(CHEMBL5180009)
Affinity DataKi:  50nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598302(CHEMBL5191079)
Affinity DataKi:  52nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598300(CHEMBL5177117)
Affinity DataKi:  53nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113283(US9695194, 8)
Affinity DataKi:  65nM ΔG°:  -42.7kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598290(CHEMBL5175954)
Affinity DataKi:  66nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50266979(CHEMBL4061897)
Affinity DataKi:  69nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in zymogen form in Pichia pastorisstrain X-33 using KHLY-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113065(US9695194, 2)
Affinity DataKi:  73nM ΔG°:  -42.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  80nM ΔG°:  -42.1kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113069(US9695194, 5)
Affinity DataKi:  85nM ΔG°:  -42.0kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598308(CHEMBL5192988)
Affinity DataKi:  90nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113248(US9695194, 7)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598289(CHEMBL5190884)
Affinity DataKi:  94nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598293(CHEMBL5172075)
Affinity DataKi:  96nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50289001(2-(2-Iodo-phenyl)-6,7-dimethoxy-benzo[d][1,3]oxazi...)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113299(US9695194, 15)
Affinity DataKi:  105nM ΔG°:  -41.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598287(CHEMBL5183937)
Affinity DataKi:  106nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113067(US9695194, 3)
Affinity DataKi:  116nM ΔG°:  -41.2kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in zymogen form in Pichia pastorisstrain X-33 using KHLY-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113295(US9695194, 12)
Affinity DataKi:  147nM ΔG°:  -40.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113300(US9695194, 16)
Affinity DataKi:  149nM ΔG°:  -40.5kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113296(US9695194, 13)
Affinity DataKi:  155nM ΔG°:  -40.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113301(US9695194, 17)
Affinity DataKi:  175nM ΔG°:  -40.1kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113297(US9695194, 14)
Affinity DataKi:  183nM ΔG°:  -40.0kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113293(US9695194, 10)
Affinity DataKi:  188nM ΔG°:  -39.9kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598304(CHEMBL5194521)
Affinity DataKi:  200nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598298(CHEMBL5206546)
Affinity DataKi:  220nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113292(US9695194, 9)
Affinity DataKi:  228nM ΔG°:  -39.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113068(US9695194, 4)
Affinity DataKi:  230nM ΔG°:  -39.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598299(CHEMBL5207509)
Affinity DataKi:  440nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50266984(CHEMBL4092637)
Affinity DataKi:  740nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in zymogen form in Pichia pastorisstrain X-33 using KHLY-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50598294(CHEMBL5185478)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK7 (30 to 253 residues) transfected in CHO cells assessed as inhibition constant using K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Queensland University Of Technology

Curated by ChEMBL
LigandPNGBDBM113294(US9695194, 11)
Affinity DataKi:  1.37E+3nM ΔG°:  -34.8kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
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