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Found 13 Enz. Inhib. hit(s) with Target = 'Methylcytosine dioxygenase TET1'
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50570893(CHEMBL4851104)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant human N-terminal Flag-tagged TET1 (1418 to 2136 residues) expressed in Baculovirus infected Sf9 cells assessed as reduction...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50570891(CHEMBL4872206)
Affinity DataIC50:  3.48E+3nMAssay Description:Inhibition of TET1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594525(CHEMBL5189434)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594530(CHEMBL5181110)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594527(CHEMBL5177921)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594520(CHEMBL5194845)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594529(CHEMBL5201158)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594528(CHEMBL5178563)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50508775(CHEMBL4457636)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of TET1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50508775(CHEMBL4457636)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of recombinant human N-terminal FLAG-tagged TET1 (1418 to 2136 residues) expressed in baculovirus infected sf9 cells assessed as reduction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594523(CHEMBL5182454)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594531(CHEMBL5198555)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethylcytosine dioxygenase TET1(Homo sapiens)
Taussig Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50594521(CHEMBL5193964)
Affinity DataIC50:  1.66E+5nMAssay Description:Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed