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Found 52 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein phosphatase PP1-gamma catalytic subunit'
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375611(CHEMBL408120)
Affinity DataKi:  3.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375608(CHEMBL406220)
Affinity DataKi:  4.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375616(CHEMBL405248)
Affinity DataKi:  8nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375613(CHEMBL261577)
Affinity DataKi:  8.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375612(CHEMBL427915)
Affinity DataKi:  17.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375609(CHEMBL406283)
Affinity DataKi:  19.6nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375614(CHEMBL259235)
Affinity DataKi:  21.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375610(CHEMBL436904)
Affinity DataKi:  23.9nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375617(CHEMBL261094)
Affinity DataKi:  32.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375615(CHEMBL261583)
Affinity DataKi:  49.7nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in E275RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D220VMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in wild typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D220VMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in E275RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in wild typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in C127SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in Y272FMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D208AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in C127SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against serine/threonine protein phosphatase 1(PP1)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  28nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type D220V by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  29nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 9PP1) mutants by natural toxins in R221SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in H248NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in R96AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  45nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in wild typeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  48nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type E275R by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  48nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in Y272FMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  58nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in R96AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  78nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type C127S by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in N124DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50177318(2-(4-(7-(4-tetradecylbenzoyl)cyclopenta[d][1,2]oxa...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against Protein phosphatase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  260nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type R96A by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50: >500nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D208AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50: >500nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in R221SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50: >500nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in H248NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50: >500nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in N124DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type Y272F by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50177316(2-(4-(7-(4-(aminomethyl)benzoyl)cyclopenta[d][1,2]...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against Protein phosphatase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50090505((1R,2S,6R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2...)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110696(4,10-Dioxa-tricyclo[5.2.1.0*2,6*]decane-3,5-dione ...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110692(7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid ...)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110695(7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid ...)
Affinity DataIC50:  4.71E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110698(7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid ...)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type D208A by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type H248N by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type N124D by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50110676(CHEMBL280487 | okadaic acid)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutant type R221S by compound was evalutadeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50177317(2-(4-(7-(4-methoxybenzoyl)cyclopenta[d][1,2]oxazin...)
Affinity DataIC50:  3.52E+4nMAssay Description:Inhibitory activity against Protein phosphatase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50090506((1R,2S,6R,7S)-5-Ethoxy-4,10-dioxa-tricyclo[5.2.1.0...)
Affinity DataIC50:  7.46E+5nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 by anhydride modified Cantharidin analoguesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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