TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 69.6nMAssay Description:Inhibition of human SGK3 using GRPRTSSFAEG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 76.5nMAssay Description:Inhibition of human SGK3 using GRPRTSSFAEG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 211nMAssay Description:Inhibition of human SGK3 in presence 500 uM presence of ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human SGK3 in presence of 500 uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGK3 using [GRPRTSSFAEG] as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human SGK3 (119 to end residues) using GRPRTSSFAEGKK as substrate incubated for 40 mins in presence of [gamma33P]ATP by rad...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of human SGK3 in presence of 500 uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 5.80nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 2.50E+3nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 96nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding constant for SGK3 kinase domainMore data for this Ligand-Target Pair