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Found 4 Enz. Inhib. hit(s) with Target = 'Threonine aspartase 1'
TargetThreonine aspartase 1(Homo sapiens (Human))
Stanford School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50300921((S)-3-((S)-2-{(S)-2-[(S)-2-((2S,3S)-2-Acetylamino-...)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThreonine aspartase 1(Homo sapiens (Human))
Stanford School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50300922((4S,7S,10S,13S,16S)-10-(3-amino-3-oxopropyl)-4-sec...)
Affinity DataIC50:  6.34E+4nMAssay Description:Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThreonine aspartase 1(Homo sapiens (Human))
Stanford School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50300923((4S,7S,10S,13S,16S)-10-(3-amino-3-oxopropyl)-4-sec...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThreonine aspartase 1(Homo sapiens (Human))
Stanford School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50300920((S)-2-((S)-2-{(S)-2-[(S)-2-((2S,3S)-2-Acetylamino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed