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Found 111 Enz. Inhib. hit(s) with Target = 'Tumor susceptibility gene 101 protein'
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362892(CHEMBL1946564)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362890(CHEMBL1946259)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362889(CHEMBL1946129)
Affinity DataKi:  8.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230460(5-[(1Z)-({[(2S,3S)-2-{[(1S)-1-{[(1S)-1-carbamoyl-3...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230449((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230470((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230450(4-carbamoyl-4-(4-carboxy-2-{[(2S,3S)-1-({1-[(2S)-2...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human Tsg101 binding to GST-tagged P6 protein by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230469((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50371256(CHEMBL1162967)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230462((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230486(5-[(1Z)-({[(3R,5S)-5-{[(1S)-1-{[(1S)-1-carbamoyl-3...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230467((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230455((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230463((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230447((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230481((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230454((4S)-4-{[(2S,3S)-3-{[(Z)-{[4-(benzyloxy)phenyl]met...)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230445((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230442((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.90E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230473((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.90E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230479((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230492((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230490((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230477((4S)-4-{[(2S,3S)-3-(aminooxy)-1-({1-[(2S)-2-[(2S,3...)
Affinity DataIC50:  2.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230483((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230464((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230457((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230448((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230485((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230451((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230482((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.50E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230487((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.50E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230475((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230465((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230444((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230466((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230493((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230446((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  2.90E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230474((4S)-4-{[(2S,4R)-4-{[(Z)-{[4-(benzyloxy)phenyl]met...)
Affinity DataIC50:  3.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230452((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230461((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  3.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230456((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  4.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230491((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  4.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230453((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  4.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230495((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  4.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230476((4S)-4-{[(2S,4R)-4-(aminooxy)-1-({1-[(2S)-2-[(2S,3...)
Affinity DataIC50:  4.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230480((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  4.80E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230484((4S)-4-{[(2S,4S)-4-{[(Z)-{[4-(benzyloxy)phenyl]met...)
Affinity DataIC50:  5.40E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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