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Found 145 Enz. Inhib. hit(s) with Target = 'Urea transporter 1'
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in human erythrocytes assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  14nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  14nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  23nMAssay Description:Inhibition of UT-B-mediated urea transport in wild type CD1 mouse erythrocytes incubated for 10 mins prior to urea addition by Stopped-flow light sca...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  25.1nMAssay Description:Reversible inhibition of mouse UT-B-mediated urea transportMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394964(CHEMBL1590659)
Affinity DataIC50:  32nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435308(CHEMBL2391344)
Affinity DataIC50:  38nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435309(CHEMBL2391345)
Affinity DataIC50:  43nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394967(CHEMBL2165784)
Affinity DataIC50:  104nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580906(CHEMBL5074722)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580917(CHEMBL5077469)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580922(CHEMBL5087071)
Affinity DataIC50:  150nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394972(CHEMBL1372659)
Affinity DataIC50:  153nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512259(CHEMBL4589155)
Affinity DataIC50:  160nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580922(CHEMBL5087071)
Affinity DataIC50:  160nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394966(CHEMBL2165785)
Affinity DataIC50:  196nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50322183(3-(4-ethylphenylsulfonyl)-N-(3-methoxypropyl)thien...)
Affinity DataIC50:  212nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512247(CHEMBL4545692)
Affinity DataIC50:  220nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512234(CHEMBL4531895)
Affinity DataIC50:  220nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512256(CHEMBL4520519)
Affinity DataIC50:  230nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580906(CHEMBL5074722)
Affinity DataIC50:  240nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512235(CHEMBL4456921)
Affinity DataIC50:  270nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580905(CHEMBL5082942)
Affinity DataIC50:  280nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435310(CHEMBL2391346)
Affinity DataIC50:  353nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580912(CHEMBL5091945)
Affinity DataIC50:  430nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394965(CHEMBL2165786)
Affinity DataIC50:  468nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512252(CHEMBL4578827)
Affinity DataIC50:  470nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580917(CHEMBL5077469)
Affinity DataIC50:  480nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580910(CHEMBL5069410)
Affinity DataIC50:  530nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394970(CHEMBL2165781)
Affinity DataIC50:  537nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512243(CHEMBL4436971)
Affinity DataIC50:  540nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580900(CHEMBL5081628)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512236(CHEMBL4535163)
Affinity DataIC50:  610nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580909(CHEMBL5084723)
Affinity DataIC50:  640nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580908(CHEMBL5083627)
Affinity DataIC50:  660nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580912(CHEMBL5091945)
Affinity DataIC50:  690nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512251(CHEMBL4526551)
Affinity DataIC50:  710nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580911(CHEMBL5075260)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435306(CHEMBL2391348)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435307(CHEMBL2391349)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435305(CHEMBL2391347)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50575413(CHEMBL4877679)
Affinity DataIC50:  800nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580916(CHEMBL5085556)
Affinity DataIC50:  810nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580905(CHEMBL5082942)
Affinity DataIC50:  840nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580913(CHEMBL5085745)
Affinity DataIC50:  870nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50512241(CHEMBL4554940)
Affinity DataIC50:  910nMAssay Description:Inhibition of urea transporter B in Sprague-Dawley rat erythrocytes incubated for 6 mins by spectrophotometric analysis based erythrocyte lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50580911(CHEMBL5075260)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50580907(CHEMBL5094101)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of rat UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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