Found 9 Enz. Inhib. hit(s) with Target = 'Acyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase'
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant Escherichia coli LpxA using UDP-GlcNAc as substrate incubated for 30 mins by spectrophotometric methodMore data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 5.00E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 3.20E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 2.20E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 4.40E+3nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 2.30E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 2.10E+3nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 1.70E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataKd: 1.20E+4nMpH: 8.0Assay Description:The fluorescence polarization assay was performed as previously described [Jenkins et al., ACS Chem. Biol., 7:1170-1177]. In 384-well black Costar pl...More data for this Ligand-Target Pair