Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with Target = 'Beta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase'
LigandPNGBDBM50117663(CHEMBL3613707)
Affinity DataIC50:  6nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117662(CHEMBL3613706)
Affinity DataIC50:  6nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117663(CHEMBL3613707)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117662(CHEMBL3613706)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50433269(CHEMBL2376303)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50:  63nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50:  63nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50:  72nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50:  79nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50:  92nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50:  100nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50433274(CHEMBL2376321)
Affinity DataIC50:  126nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50:  204nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50:  205nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117666(CHEMBL3613710)
Affinity DataIC50:  365nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50:  389nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50:  394nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50433272(CHEMBL2376325)
Affinity DataIC50:  398nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117666(CHEMBL3613710)
Affinity DataIC50:  398nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117664(CHEMBL3613708)
Affinity DataIC50:  597nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117659(CHEMBL3613703)
Affinity DataIC50:  631nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117664(CHEMBL3613708)
Affinity DataIC50:  631nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117659(CHEMBL3613703)
Affinity DataIC50:  682nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50:  760nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50:  794nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM201239(US9187424, 6-2)
Affinity DataIC50: >820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50579519(CHEMBL3912712)
Affinity DataIC50: >820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50579526(CHEMBL4878564)
Affinity DataIC50: >820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50433273(CHEMBL2376322)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117660(CHEMBL3613704)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117660(CHEMBL3613704)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117661(CHEMBL3613705)
Affinity DataIC50:  3.84E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117661(CHEMBL3613705)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090510(CHEMBL3581716)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of full length human MGAT3 transfected in Sf-21 cells using [1-14C]oleoyl-CoA assessed as incorporation of radioactivity into lip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM276750((S)-2-(5-((3-ethoxypyridin-2-yl)oxy)pyridin-3-yl)-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human MGAT3 using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates assessed as incorporation of [1-14C]decanoyl into di...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM276748(US10071992, Example 3.5 | US10071992, Example 5 | ...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human MGAT3 using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates assessed as incorporation of [1-14C]decanoyl into di...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed