Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with Target = 'Macrophage inflammatory protein-1 alpha receptor'
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445006(CHEMBL3099943)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210979((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  17nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210977((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  20nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210982((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  21nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210971((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  24nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210970((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  49nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445005(CHEMBL3099944)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445004(CHEMBL3099945)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50208999((R)-1-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  59nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435676(CHEMBL2391938)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210972((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  87nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445003(CHEMBL3099946)
Affinity DataIC50:  90nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445002(CHEMBL3099947)
Affinity DataIC50:  101nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435673(CHEMBL2391795)
Affinity DataIC50:  114nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50210976((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50:  130nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435671(CHEMBL2391793)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445008(CHEMBL3099941)
Affinity DataIC50:  447nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435690(CHEMBL2391803)
Affinity DataIC50:  880nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435684(CHEMBL2391794)
Affinity DataIC50:  890nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435669(CHEMBL2391809)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50444998(CHEMBL3099951)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445001(CHEMBL3099948)
Affinity DataIC50:  1.58E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50444999(CHEMBL3099950)
Affinity DataIC50:  1.62E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445007(CHEMBL3099942)
Affinity DataIC50:  1.76E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50444989(CHEMBL3099960)
Affinity DataIC50:  1.78E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50445000(CHEMBL3099949)
Affinity DataIC50:  2.11E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435668(CHEMBL2391800)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50444995(CHEMBL3099954)
Affinity DataIC50: >6.00E+3nMAssay Description:Displacement of [125I]MIP-1alpha from rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435666(CHEMBL2391804)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50435667(CHEMBL2391796)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at rat CCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rattus norvegicus)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50399208(CHEMBL2180528)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in rat thioglycolate-elicited peritoneal cells incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed