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Found 227 Enz. Inhib. hit(s) with Target = 'Cytosol aminopeptidase'
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50024594((R)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50316049(1-amino-3-phenylpropylphosphonic acid | CHEMBL1090...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025048(CHEMBL3355099)
Affinity DataKi:  5nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50078125((1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025043(CHEMBL3355104)
Affinity DataKi:  20nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [435-519](Sus scrofa)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50022748(2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349)
Affinity DataKi:  22nMAssay Description:Competitive inhibition of LAP in porcine kidney microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  30nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025041(CHEMBL3355106)
Affinity DataKi:  39nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50225458((2S)-3-[(R)-[(1S)-1-amino-3-phenylpropyl](hydroxy)...)
Affinity DataKi:  45nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025042(CHEMBL3355105)
Affinity DataKi:  50nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataKi:  50nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129685(2-Amino-4-methyl-pentanal | CHEMBL88476)
Affinity DataKi:  60nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  65nMAssay Description:Inhibition of LAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190111(CHEMBL327844)
Affinity DataKi:  66nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025070(CHEMBL3355110)
Affinity DataKi:  74nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)
Affinity DataKi:  74nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50089610((Z)-(S)-5-Amino-7-methyl-4-oxo-oct-2-enoic acid me...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity of the compound against leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025099(CHEMBL3355111)
Affinity DataKi:  108nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50027041(2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...)
Affinity DataKi:  120nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025066(CHEMBL3355109)
Affinity DataKi:  138nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025044(CHEMBL3355103)
Affinity DataKi:  157nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025050(CHEMBL3355108)
Affinity DataKi:  195nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  200nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50337147((RS)-1-amino-3-cyclohexylpropylphosphonic acid | C...)
Affinity DataKi:  210nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025047(CHEMBL3355100)
Affinity DataKi:  213nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50025046(CHEMBL3355101)
Affinity DataKi:  215nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [33-68,L62W](Sus scrofa (Pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50024597((S)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...)
Affinity DataKi:  220nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  220nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  230nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024594((R)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...)
Affinity DataKi:  230nMAssay Description:Inhibition of Leucine aminopeptidase isolated from porcine kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316047(1-amino-2-methylbutylphosphonic acid monophenylest...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50234656((R)-3-[((R)-1-amino-3-phenyl-propyl)-hydroxy-phosp...)
Affinity DataKi:  271nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)
Affinity DataKi:  330nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50022747(2-(3-Amino-2-hydroxy-4-phenyl-thiobutyrylamino)-4-...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024596((R)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  420nMAssay Description:Inhibition of Leucine aminopeptidase isolated from porcine kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316048(1-amino-2-phenylethylphosphonic acid monophenyl es...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024592((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024590(1-Ammonium-octane-1-phosphonic acid anion | CHEMBL...)
Affinity DataKi:  470nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Universit£

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of bovine LAPc using L-leucine-p-nitroanilide as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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