Found 7 Enz. Inhib. hit(s) with Target = '4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5'
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataKi: 6.71E+4nMAssay Description:Inhibition of Fucosyltransferase 5 by the compound was evaluated; Competitive inhibitionMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataKi: 8.89E+5nMAssay Description:Inhibition of Fucosyltransferase 5 by the compound was evaluated; Weak competitive inhibitionMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of GnRH-stimulated luteinizing hormone (LH) release in rat pituitary cellsMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
University Of California Los Angeles
Curated by ChEMBL
University Of California Los Angeles
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair