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Found 2 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase SETD1B'
TargetHistone-lysine N-methyltransferase SETD1B(Homo sapiens)
The Walter And Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50524882(CHEMBL4465202)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of C-terminal GST-tagged human SET1B (1629 to 1923 amino acids) expressed in Escherichia coli using core histone as substrate in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase SETD1B(Homo sapiens)
The Walter And Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50508569(CHEMBL4557353)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of SETD1B (unknown origin) using SAM as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by Alpha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed