Compile Data Set for Download or QSAR
maximum 50k data
Found 925 Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1'
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121307(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  0.560nM ΔG°:  -54.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121274(US8722896, (+/-)-4-(Indol-7-ylmethyl)-N-(9- chloro...)
Affinity DataKi:  1.13nM ΔG°:  -53.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121324(US8722896, (-)-(2R)-2-Methyl-3-((3- hydroxy)benzyl...)
Affinity DataKi:  1.15nM ΔG°:  -53.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121105(US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (9-chl...)
Affinity DataKi:  1.22nM ΔG°:  -52.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463303((-)-(2R)-1-(2-Methoxybenzyl)- N-(9-chloro-3,4-dihy...)
Affinity DataKi:  1.49nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121307(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  1.56nM ΔG°:  -52.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121105(US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (9-chl...)
Affinity DataKi:  1.98nM ΔG°:  -51.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121202(US8722896, (+)-(2S)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  2.38nM ΔG°:  -51.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463304((-)-(2R)-1-(3-Methoxybenzyl)- N-(9-chloro-3,4-dihy...)
Affinity DataKi:  2.5nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463306((-)-(2R)-1-(4-Fluoro-3- methoxybenzyl)-N-(9-chloro...)
Affinity DataKi:  2.60nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463307((-)-(3R)-1-(benzimidazol-4- ylmethyl)-N-(9-chloro-...)
Affinity DataKi:  2.60nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121116(US8722896, (-)-(3R)-N-(9-chloro-3,4- dihydro-2H-1,...)
Affinity DataKi:  2.82nM ΔG°:  -50.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121259(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  3.29nM ΔG°:  -50.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463308((-)-(2R)-2-Methyl-3- (benzimidazol-4- ylmethylamin...)
Affinity DataKi:  3.5nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121046(US8722896, (-)-(3R)-1-(1-Methyl-indol-4- ylmethyl)...)
Affinity DataKi:  3.64nM ΔG°:  -50.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121294(US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (9-chl...)
Affinity DataKi:  3.68nM ΔG°:  -50.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121261(US8722896, (-)-(3R)-1-(N-methyl-indol-4- ylmethyl)...)
Affinity DataKi:  3.74nM ΔG°:  -50.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121157(US8722896, (+/-)-2-Methyl-3-(2,3-dihydro-1- benzof...)
Affinity DataKi:  3.78nM ΔG°:  -50.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121319(US8722896, (+/-)-2-Methyl-3-((3- acetoxy)benzylami...)
Affinity DataKi:  3.84nM ΔG°:  -50.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121088(US8722896, (-)-(3R)-1-(3-Methoxybenzyl)- N-(9-chlo...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121290(US8722896, (+/-)-(3R)-4-(Indol-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  4.02nM ΔG°:  -49.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121202(US8722896, (+)-(2S)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  4.08nM ΔG°:  -49.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463321((-)-(2R)-1-(4,6-Difluoro-3- methoxybenzyl)-N-(9-ch...)
Affinity DataKi:  4.09nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121202(US8722896, (+)-(2S)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  4.24nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121261(US8722896, (-)-(3R)-1-(N-methyl-indol-4- ylmethyl)...)
Affinity DataKi:  4.26nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463326((+-)-2-Methyl-3-((3-hydroxy-4- fluoro)benzylamino)...)
Affinity DataKi:  4.40nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121299(US8722896, (+/-)-2-Methyl-3-(N-methyl-indol- 4-ylm...)
Affinity DataKi:  4.5nM ΔG°:  -49.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121310(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  4.60nM ΔG°:  -49.5kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121106(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  4.70nM ΔG°:  -49.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121313(US8722896, (+/-)-2-Methyl-3-(2,3- dimethylbenzylme...)
Affinity DataKi:  4.70nM ΔG°:  -49.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121300(US8722896, (-)-(3R)-1-(N-methyl-indol-4- ylmethyl)...)
Affinity DataKi:  4.72nM ΔG°:  -49.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121303(US8722896, (+/-)-2-Methyl-3-(N-methyl-indol- 7-ylm...)
Affinity DataKi:  4.74nM ΔG°:  -49.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121277(US8722896, (+/-)-4-(Indolin-4-ylmethyl)-N-(9- chlo...)
Affinity DataKi:  4.80nM ΔG°:  -49.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121205(US8722896, (+)-(2S)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  4.90nM ΔG°:  -49.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121086(US8722896, (-)-(3R)-1-(3-Hydroxybenzyl)- N-(9-chlo...)
Affinity DataKi:  5.20nM ΔG°:  -49.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121116(US8722896, (-)-(3R)-N-(9-chloro-3,4- dihydro-2H-1,...)
Affinity DataKi:  5.34nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121274(US8722896, (+/-)-4-(Indol-7-ylmethyl)-N-(9- chloro...)
Affinity DataKi:  5.40nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121281(US8722896, (+/-)-4-(2,3-Dihydro-1- benzofuran-7-yl...)
Affinity DataKi:  5.46nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121321(US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)- N-(9-chl...)
Affinity DataKi:  5.5nM ΔG°:  -49.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463309((+-)-2-Methyl-3-(benzimidazol- 4-ylmethylamino)-N-...)
Affinity DataKi:  5.60nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121262(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
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TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463313((-)-(2R)-1-(5-fluro- benzimidazol-4-ylmethyl)-N- (...)
Affinity DataKi:  6.14nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM463316((-)-(3R)-1-(4,6-Difluoro-3- methoxybenzyl)-N-(9-ch...)
Affinity DataKi:  6.14nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121046(US8722896, (-)-(3R)-1-(1-Methyl-indol-4- ylmethyl)...)
Affinity DataKi:  6.5nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121292(US8722896, (+/-)-(3R)-4-(Indol-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  6.62nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
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TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121253(US8722896, (-)-(2R)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  6.68nM ΔG°:  -48.5kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121205(US8722896, (+)-(2S)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  6.96nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121086(US8722896, (-)-(3R)-1-(3-Hydroxybenzyl)- N-(9-chlo...)
Affinity DataKi:  7.10nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121202(US8722896, (+)-(2S)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  7.18nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121145(US8722896, (+/-)-2-Methyl-3-((2- methoxybenzyl)met...)
Affinity DataKi:  7.26nM ΔG°:  -48.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
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