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Found 33 Enz. Inhib. hit(s) with Target = 'Protein S100-B'
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429682(CHEMBL2335383)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429681(CHEMBL2094307 | DNDI1416906)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429679(CHEMBL2335386)
Affinity DataKi:  1.75E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429680(CHEMBL2335384)
Affinity DataKi:  2.51E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM34166((2,4-dipiperidinophenyl)amine | 2,4-Di-piperidin-1...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146593(CHEMBL3764851)
Affinity DataIC50:  6.70E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429682(CHEMBL2335383)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429681(CHEMBL2094307 | DNDI1416906)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146592(CHEMBL3764285)
Affinity DataIC50:  1.83E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429679(CHEMBL2335386)
Affinity DataIC50:  2.28E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429680(CHEMBL2335384)
Affinity DataIC50:  3.15E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429684(4-(4-Methoxybenzylideneamino)Phenol | CHEMBL67238)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50429683(4-((4-(Phenylamino)Phenylimino)Methyl)Phenol | CHE...)
Affinity DataIC50:  4.21E+4nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146595(CHEMBL3765382)
Affinity DataIC50:  5.11E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50100895(2-(4-(4-carbamimidoylphenoxy)phenyl)-1H-indole-6-c...)
Affinity DataIC50:  6.66E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human S100B/human TAMRA-p53(367-388) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146596(CHEMBL3765054)
Affinity DataIC50:  9.82E+5nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146594(CHEMBL3765771)
Affinity DataIC50:  2.22E+6nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146594(CHEMBL3765771)
Affinity DataKd:  2.03E+5nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146595(CHEMBL3765382)
Affinity DataKd:  4.60E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146593(CHEMBL3764851)
Affinity DataKd:  500nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146592(CHEMBL3764285)
Affinity DataKd:  1.60E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50146596(CHEMBL3765054)
Affinity DataKd:  8.95E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50100895(2-(4-(4-carbamimidoylphenoxy)phenyl)-1H-indole-6-c...)
Affinity DataKd:  6.00E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to recombinant rat calcium loaded S100-B by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetProtein S100-B(Rattus norvegicus)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataKd:  4.40E+4nMAssay Description:Binding affinity to recombinant rat calcium loaded S100-B by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154226(5-{[1,3-Dioxo-2-(2,4,6-trimethyl-phenyl)-2,3-dihyd...)
Affinity DataKd:  1.20E+5nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154225(2-(3-tert-Butylcarbamoyl-phenyl)-1,3-dioxo-2,3-dih...)
Affinity DataKd:  8.10E+3nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154224(CHEMBL434915 | N-[4-(1,5-Dimethyl-3-oxo-2-phenyl-2...)
Affinity DataKd:  4.50E+3nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154222(1-[amino(iminiumyl)methyl]-3-(2-benzoyl-4-chloroph...)
Affinity DataKd:  4.50E+3nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154221(5-((2E)-2-{[5-(3-carboxy-4-chlorophenyl)-2-furyl]m...)
Affinity DataKd:  1.83E+4nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein S100-B(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50154223(CHEMBL185802 | N-(2,3-dichlorophenyl)imidodicarbon...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding to holo-S100B proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed