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Found 8 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1C1'
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50225220(CHEMBL559 | D-thyroxine | O-(4-hydroxy-3,5-diiodop...)
Affinity DataKi:  270nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103763(CHEBI:11684 | REVERSE TRIIODOTHYRONINE | Reverse T...)
Affinity DataKi:  910nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM18862(2-[4-(4-hydroxy-3-iodophenoxy)-3,5-diiodophenyl]ac...)
Affinity DataKi:  2.15E+3nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM18860((2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-di...)
Affinity DataKi:  2.42E+4nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50366524(ESTRONE | ESTROPIPATE | Estrone 3-sulfate | Estron...)
Affinity DataKi:  5.31E+4nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50344959(17beta-Estradiol-17-(beta-D-glucuronide) | CHEMBL1...)
Affinity DataKi: >1.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)
Affinity DataKi:  1.09E+5nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50206509(4-Dipropylsulfamoyl-benzoic acid | 4-Dipropylsulfa...)
Affinity DataKi:  2.93E+5nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed