Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 460nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 900nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.90E+3nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 7.10E+3nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 8.00E+3nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 8.20E+3nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.21E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.38E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.60E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 2.19E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 3.20E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 4.69E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 6.52E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 6.90E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 7.74E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 9.28E+4nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.02E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.05E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 1.75E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 3.05E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: 3.57E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1 [C171Q](Mycobacterium tuberculosis)
University Of Wuerzburg
University Of Wuerzburg
Affinity DataKi: 3.84E+5nMpH: 8.5Assay Description:Binding of TLM18 to wild-type and mutant KasA was quantified by monitoring changes in the intrinsic tryptophan fluorescence of the enzyme at waveleng...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Institute For Chemical Biology & Drug Discovery
Institute For Chemical Biology & Drug Discovery
Affinity DataKi: >4.00E+5nMpH: 8.5Assay Description:Binding of TLM and the TLM analogs to KasA was quantified by monitoring changes in the intrinsic tryptophan fluroescence of the enzyme using 280-nm e...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
Universidad Aut£Noma De Nuevo Le£N
Curated by ChEMBL
Universidad Aut£Noma De Nuevo Le£N
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv Fab1More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair