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Found 31 Enz. Inhib. hit(s) with Target = 'D-alanine--D-alanine ligase'
TargetD-alanine--D-alanine ligase(Helicobacter pylori (strain HPAG1))TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKi:  4.30E+3nMAssay Description:Competitive inhibition of Helicobacter pylori Ddl using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase(Helicobacter pylori (strain HPAG1))TBA
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  3.10E+4nMAssay Description:Competitive inhibition of Helicobacter pylori Ddl using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520701(CHEMBL4515707)
Affinity DataIC50:  100nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520694(CHEMBL4535288)
Affinity DataIC50:  370nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520691(CHEMBL4457124)
Affinity DataIC50:  510nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520692(CHEMBL4441028)
Affinity DataIC50:  520nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520690(CHEMBL4547125)
Affinity DataIC50:  550nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520695(CHEMBL4450059)
Affinity DataIC50:  560nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520684(CHEMBL4566999)
Affinity DataIC50:  580nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520687(CHEMBL4445254)
Affinity DataIC50:  630nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520700(CHEMBL4448556)
Affinity DataIC50:  700nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520696(CHEMBL4524762)
Affinity DataIC50:  710nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520693(CHEMBL4591078)
Affinity DataIC50:  730nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520698(CHEMBL4472847)
Affinity DataIC50:  790nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50133806(CHEMBL3633780)
Affinity DataIC50:  800nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520703(CHEMBL4594055)
Affinity DataIC50:  830nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520689(CHEMBL4531935)
Affinity DataIC50:  840nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520685(CHEMBL4461445)
Affinity DataIC50:  930nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520699(CHEMBL4514663)
Affinity DataIC50:  930nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520688(CHEMBL4453039)
Affinity DataIC50:  970nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520697(CHEMBL4465913)
Affinity DataIC50:  990nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520702(CHEMBL4451238)
Affinity DataIC50:  990nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520683(CHEMBL4476621)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase B(Escherichia coli K-12)TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.99E+4nMAssay Description:Competitive inhibition of Escherichia coli DdlB using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase(Helicobacter pylori (strain HPAG1))TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  4.85E+4nMAssay Description:Competitive inhibition of Helicobacter pylori Ddl using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase(Helicobacter pylori (strain HPAG1))TBA
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.33E+5nMAssay Description:Competitive inhibition of Helicobacter pylori Ddl using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase B(Escherichia coli K-12)TBA
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.63E+5nMAssay Description:Competitive inhibition of Escherichia coli DdlB using ATP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD-alanine--D-alanine ligase B(Escherichia coli K-12)TBA
LigandPNGBDBM50589509(CHEMBL5173242)
Affinity DataIC50:  2.43E+5nMAssay Description:Inhibition of recombinant Escherichia coli DdlB using D-alanine as substrate incubated for 20 mins and measured by malachite green based colorimetric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50103516(CHEBI:40009 | Cycloserine | Seromycin)
Affinity DataIC50:  2.62E+5nMAssay Description:Inhibition of Enterococcus faecalis JH2-2 C-terminal 6His-tagged DdlB expressed in Escherichia coli LMG194 preincubated for 30 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Enterococcus faecalis (strain ATCC 700802 / V583))
Universit£

Curated by ChEMBL
LigandPNGBDBM50520686(CHEMBL4537639)
Affinity DataIC50:  4.32E+5nMAssay Description:Inhibition of Enterococcus faecalis DdlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-alanine--D-alanine ligase(Helicobacter pylori (strain HPAG1))TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKd:  1.29E+4nMAssay Description:Binding affinity to Helicobacter pylori Ddl by surface plasmon resonance biosensor technologyMore data for this Ligand-Target Pair
In DepthDetails Article