Compile Data Set for Download or QSAR
maximum 50k data
Found 130 Enz. Inhib. hit(s) with Target = 'Disks large homolog 4'
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(CHEMBL493688 | N-Cyclohexylethyl-ETAV)
Affinity DataKi:  450nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(CHEMBL493688 | N-Cyclohexylethyl-ETAV)
Affinity DataKi:  630nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339567((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cyclohexyl-8...)
Affinity DataKi:  630nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339545((4S,7S,10S,13S)-4-(2-carboxyethyl)-10-(carboxymeth...)
Affinity DataKi:  750nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(CHEMBL493688 | N-Cyclohexylethyl-ETAV)
Affinity DataKi:  940nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252828(CHEMBL493689 | N-(Naphthalene-2-yl)ethyl-ETAV)
Affinity DataKi:  950nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV)
Affinity DataKi:  980nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252828(CHEMBL493689 | N-(Naphthalene-2-yl)ethyl-ETAV)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339569((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252826(CHEMBL494486 | N-Cyclohexylmethyl-ETAV)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339568((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339548((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339555((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cycloheptyl-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339552((3S,6S,9S,12S)-1-(bicyclo[2.2.1]heptan-2-yl)-3-(2-...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252826(CHEMBL494486 | N-Cyclohexylmethyl-ETAV)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339554((3S,6S,9S,12S)-3-(2-carboxyethyl)-1-cycloheptyl-6-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339553((2S,5S,8S,11S)-14-(bicyclo[2.2.1]heptan-2-yl)-11-(...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252715(CHEMBL494895 | N-Phenylethyl-ETAV)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339556((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339547((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253144(CHEMBL505051 | KSG-LDTKNYKQTSV)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252752(CHEMBL495099 | N-Phenylpropyl-ETAV)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339551((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252713(CHEMBL492642 | FETAV)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252752(CHEMBL495099 | N-Phenylpropyl-ETAV)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339539((4S,7S,10S,13S)-10-(carboxymethyl)-1-cyclohexyl-7-...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252825(CHEMBL494485 | N-Butyl-ETAV)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253143(CHEMBL445253 | KSG-YEKLSSIESDV)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252824(CHEMBL494287 | N-Propyl-ETAV)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339557((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339546((4S,7S,10S,13S)-4-(3-amino-3-oxopropyl)-10-(carbox...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253145(CHEMBL502630 | YGRKKRRQRRR-KLSSIESDV)
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252715(CHEMBL494895 | N-Phenylethyl-ETAV)
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253145(CHEMBL502630 | YGRKKRRQRRR-KLSSIESDV)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339558((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252714(CHEMBL492643 | N-Benzyl-ETAV)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252713(CHEMBL492642 | FETAV)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV)
Affinity DataKi:  6.70E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339551((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253143(CHEMBL445253 | KSG-YEKLSSIESDV)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1-2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252824(CHEMBL494287 | N-Propyl-ETAV)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252714(CHEMBL492643 | N-Benzyl-ETAV)
Affinity DataKi:  7.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV)
Affinity DataKi:  7.80E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339538((4S,7S,10S,13S)-1-cyclohexyl-7-((R)-1-hydroxyethyl...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339569((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252825(CHEMBL494485 | N-Butyl-ETAV)
Affinity DataKi:  8.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339556((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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