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Found 150 Enz. Inhib. hit(s) with Target = 'Elongation of very long chain fatty acids protein 6'
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of ELOVL6 in mouse H2.35 cells assessed as elongation indexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299964(4-Fluoro-N-{[2-oxo-6-(1H-pyrazol-5-yl)-4-(trifluor...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249891(3-[2-(4-methyllphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249844(3-[2-(4-isopropylphenyl)-5-methyl-3-oxo-2,3-dihydr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249791(3-[2-(4-chlorophenyl)-5-methyl-3-oxo-2,3-dihydro-1...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249843(3-[2-(4-cyanophenyl)-5-methyl-3-oxo-2,3-dihydro-1H...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249815(3-[2-(4-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299963(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-4-yl)-4-(trif...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299963(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-4-yl)-4-(trif...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299963(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-4-yl)-4-(trif...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299948(CHEMBL572158 | N-{[(+)-6-Chloro-2-oxo-4-(trifluoro...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299965(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-1-yl)-4-(trif...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299948(CHEMBL572158 | N-{[(+)-6-Chloro-2-oxo-4-(trifluoro...)
Affinity DataIC50:  26nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299948(CHEMBL572158 | N-{[(+)-6-Chloro-2-oxo-4-(trifluoro...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299965(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-1-yl)-4-(trif...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299965(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-1-yl)-4-(trif...)
Affinity DataIC50:  29nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ELOVL6 in mouse H2.35 cells assessed as reduction in elongation index using [14C]palmitic acid as radiotracer after 4 hrs by radio-HPLC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299946(1-{[(-)-6-Chloro-2-oxo-4-(trifluoromethyl)-1,4-dih...)
Affinity DataIC50:  31nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50:  31nMAssay Description:Inhibition of mouse ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293790(CHEMBL550828 | N-(4-Isopropylphenyl)-3-endo-(pheny...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299946(1-{[(-)-6-Chloro-2-oxo-4-(trifluoromethyl)-1,4-dih...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299946(1-{[(-)-6-Chloro-2-oxo-4-(trifluoromethyl)-1,4-dih...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299951(CHEMBL582825 | N-{[6-Chloro-2-oxo-4-(trifluorometh...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299969(4-Fluoro-N-{[2-oxo-6-(2-oxopyrrolidin-1-yl)-4-(tri...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249814(3-[2-(3-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249842(3-[2-(4-fluorophenyl)-5-methyl-3-oxo-2,3-dihydro-1...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249790(3-[2-(3-chlorophenyl)-5-methyl-3-oxo-2,3-dihydro-1...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299963(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-4-yl)-4-(trif...)
Affinity DataIC50:  50nMAssay Description:Inhibition of ELOVL6 in mouse H2.35 cells assessed as elongation indexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299965(4-Fluoro-N-{[(+)-2-oxo-6-(1H-pyrazol-1-yl)-4-(trif...)
Affinity DataIC50:  58nMAssay Description:Inhibition of ELOVL6 in mouse H2.35 cells assessed as elongation indexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249813(3-[2-(2-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298994((1R*,4S*,6R*)-(+/-)-N-[4-(Propan-2-yloxy)phenyl]-2...)
Affinity DataIC50:  67nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299970(4-Fluoro-N-{[2-oxo-6-(2-oxo-1,3-oxazolidin-3-yl)-4...)
Affinity DataIC50:  67nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298985((1R*,4S*,6R*)-(+/-)-2-(Phenylsulfonyl)-N-[4-(propa...)
Affinity DataIC50:  70nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50:  73nMAssay Description:Inhibition of C-terminal V5-epitope-tagged mouse ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50378036(CHEMBL1163008)
Affinity DataIC50:  78nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50:  79nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298967((1R*,4S*,6R*)-(+/-)-N-[4-(Propan-2-yloxy)phenyl]-2...)
Affinity DataIC50:  80nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50:  94nMAssay Description:Inhibition of mouse ELOVL6 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299959(4-Fluoro-N-{[2-oxo-4-(trifluoromethyl)-1,4-dihydro...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299966(4-Fluoro-N-{[2-oxo-6-(1H-1,2,4-triazol-5-yl)-4-(tr...)
Affinity DataIC50:  97nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249713(3-(5-ethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299961(4-Fluoro-N-{[2-oxo-6-(2-oxopyridin-1(2H)-yl)-4-(tr...)
Affinity DataIC50:  106nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298991((1R*,4S*,6R*)-(+/-)-2-[(3-Fluorophenyl)sulfonyl]-N...)
Affinity DataIC50:  110nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298969((1R*,4S*,6R*)-(+/-)-N-[4-(Propan-2-yloxy)phenyl]-2...)
Affinity DataIC50:  120nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298971((1R*,4S*,6R*)-(+/-)-2-(Butylsulfonyl)-N-[4-(propan...)
Affinity DataIC50:  120nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299962(4-Fluoro-N-{[6-(isoxazol-4-yl)-2-oxo-4-(trifluorom...)
Affinity DataIC50:  121nMAssay Description:Inhibition of human ELOVL6 expressed in Pichia pastoris using palmitoyl-CoA by long chain fatty acyl-CoA elongation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 6(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249764(3'-(5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human ELOVL6 expressed in african green monkey COS7 cells assessed as palmitoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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