Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with Target = 'Gastrotropin'
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534537(CHEMBL4576559)
Affinity DataKd:  2.90E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534538(CHEMBL4439741)
Affinity DataKd:  4.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM14324(5,6-dimethyl-1H-1,3-benzodiazol-2-amine | Fragment...)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by 2 site binding model based surf...More data for this Ligand-Target Pair
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534542(CHEMBL391815)
Affinity DataKd:  3.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534540(CHEMBL4532670)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534539(CHEMBL4454723)
Affinity DataKd:  8.00E+4nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataKd:  2.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM14324(5,6-dimethyl-1H-1,3-benzodiazol-2-amine | Fragment...)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534544(CHEMBL4587123)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534541(CHEMBL4454549)
Affinity DataKd:  3.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50383377(CHEMBL2030560 | US10544104, Compound 92 | US976503...)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM14324(5,6-dimethyl-1H-1,3-benzodiazol-2-amine | Fragment...)
Affinity DataKd:  2.94E+4nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by 1 site binding model based surf...More data for this Ligand-Target Pair
TargetGastrotropin(Homo sapiens)
Takeda Cambridge

Curated by ChEMBL
LigandPNGBDBM50534543(CHEMBL4555681)
Affinity DataKd:  4.00E+4nMAssay Description:Binding affinity to recombinant human N-terminal His6 and Avi-tagged FABP6 expressed in Escherichia coli NEB cells by surface plasmon resonance metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed