Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = '1-alkyl-2-acetylglycerophosphocholine esterase'
Target1-alkyl-2-acetylglycerophosphocholine esterase(Sus scrofa)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-(ethylamino)hexadecan-1-ol | 2-Ethylamino-hexade...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-alkyl-2-acetylglycerophosphocholine esterase(Sus scrofa)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-alkyl-2-acetylglycerophosphocholine esterase(Sus scrofa)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50:  4.10E+3nMAssay Description:Compound was tested for its ability to inhibit porcine pancreas phospholipase-A2More data for this Ligand-Target Pair
In DepthDetails Article