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Found 777 Enz. Inhib. hit(s) with Target = 'Glycogen phosphorylase, liver form'
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50148913(CHEMBL3770455)
Affinity DataKi:  26nMAssay Description:Competitive inhibition of His6-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inorg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50241632(CHEMBL4101331)
Affinity DataKi:  143nMAssay Description:Competitive inhibition of 6xHis-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50148915(CHEMBL3770514)
Affinity DataKi:  156nMAssay Description:Competitive inhibition of His6-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inorg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50437354(CHEMBL2408225)
Affinity DataKi:  172nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50437354(CHEMBL2408225)
Affinity DataKi:  172nMAssay Description:Competitive inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using varying levels of glucose-1-phosphate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50016703(2-Hydroxymethyl-pyrrolidine-3,4-diol | BDBM5003148...)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against pig Liver glycogen phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50437355(CHEMBL2408224)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50437355(CHEMBL2408224)
Affinity DataKi:  1.35E+3nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50312361(CHEMBL4169281)
Affinity DataKi:  2.02E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50312362(CHEMBL4176460)
Affinity DataKi:  2.23E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50313014(CHEMBL4172670)
Affinity DataKi:  2.67E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50241633(CHEMBL4095486)
Affinity DataKi:  2.73E+3nMAssay Description:Competitive inhibition of 6xHis-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50538946(CHEMBL4646575)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50312225(CHEMBL4161353)
Affinity DataKi:  3.88E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50211296((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-6...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50211294((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-2...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50241634(CHEMBL4068103)
Affinity DataKi:  7.60E+3nMAssay Description:Competitive inhibition of 6xHis-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50312632(CHEMBL4164542)
Affinity DataKi:  8.91E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using glucose-1-phosphate as substrate in presence of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  1.09E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50211289(5-[4-(6,7-dibromo-2,3-dihydrobenzo[1,4]dioxin-2-yl...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50215446(CHEMBL3351144)
Affinity DataKi:  1.28E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50215446(CHEMBL3351144)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50215446(CHEMBL3351144)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase a in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50538945(CHEMBL4638064)
Affinity DataKi:  2.59E+4nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50211294((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-2...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibition of rat liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibition of rat liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase a in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University

Curated by ChEMBL
LigandPNGBDBM50211294((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-2...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibition of rat liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50211288(5-[4-(6,7-dibromo-2,3-dihydrobenzo[1,4]dioxin-2-yl...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50241635(CHEMBL4087784)
Affinity DataKi:  3.08E+4nMAssay Description:Competitive inhibition of 6xHis-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50538948(CHEMBL4648992)
Affinity DataKi:  4.36E+4nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50148917(CHEMBL3770888)
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50211286(5-[4-(6-bromo-2,3-dihydrobenzo[1,4]dioxin-2-ylmeth...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50538949(CHEMBL4640451)
Affinity DataKi:  1.34E+5nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50538947(CHEMBL4642474)
Affinity DataKi:  1.72E+5nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50148914(CHEMBL3769528)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition of human liver GPa using Glc-1-P as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  4.28E+6nMAssay Description:Competitive inhibition of His6-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inorg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  4.90E+6nMAssay Description:Inhibition of glycogen phosphorylase a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135554(4-{3-[(4-Nitro-pyridine-2-carbonyl)-amino]-naphtha...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135558(4-{3-Fluoro-2-[(4-nitro-pyridine-2-carbonyl)-amino...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135553(4-{3-[(4-Chloro-pyridine-2-carbonyl)-amino]-naphth...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135565(4-{3-[(4-Methoxy-pyridine-2-carbonyl)-amino]-napht...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50133440(1-(4-Chloro-benzyl)-4-(2-chloro-phenyl)-6-methyl-1...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM24393(2,3-dichloro-N-{1-[(2R)-2,3-dihydroxypropyl]-2-oxo...)
Affinity DataIC50:  2nMAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135562(4-{2-[(4-Nitro-pyridine-2-carbonyl)-amino]-phenoxy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM27730((2S,3R)-3-(tert-butoxy)-2-{[4-(4-methoxyphenyl)-2-...)
Affinity DataIC50:  3nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM27747((2S,3R)-3-(tert-butoxy)-2-{[2-({[4-(cyclopropylmet...)
Affinity DataIC50:  3nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50135557(4-{3-[(4-Ethyl-pyridine-2-carbonyl)-amino]-naphtha...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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