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Found 564 Enz. Inhib. hit(s) with Target = 'Period circadian protein homolog 2'
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50140894(CHEMBL3754467 | US10383880, Example 124)
Affinity DataEC50:  726nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50140895(CHEMBL3753417 | US10383880, Example 4)
Affinity DataEC50:  1.09E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140896(CHEMBL3752727 | US10383880, Example 14)
Affinity DataEC50:  415nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140904(CHEMBL3752018 | US10383880, Example 113)
Affinity DataEC50:  479nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140907(CHEMBL1487843 | US10383880, Example 32)
Affinity DataEC50:  781nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140915(CHEMBL3754372 | US10383880, Example 45)
Affinity DataEC50:  505nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140918(CHEMBL3752371)
Affinity DataEC50:  408nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140919(CHEMBL3753078 | US10383880, Example 46)
Affinity DataEC50:  511nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140920(CHEMBL3752323 | US10383880, Example 49)
Affinity DataEC50:  178nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140921(CHEMBL3753693 | US10383880, Example 56)
Affinity DataEC50:  446nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140922(CHEMBL3752819 | US10383880, Example 57)
Affinity DataEC50:  129nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140692(CHEMBL3754517 | US10383880, Example 84)
Affinity DataEC50:  1.00E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140693(CHEMBL3753394 | US10383880, Example 11)
Affinity DataEC50:  288nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140696(CHEMBL3752613 | US10383880, Example 16)
Affinity DataEC50:  557nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140697(CHEMBL3754783)
Affinity DataEC50:  374nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140698(CHEMBL3753223 | US10383880, Example 13)
Affinity DataEC50:  361nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140700(CHEMBL3754797 | US10383880, Example 85)
Affinity DataEC50:  1.18E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140701(CHEMBL3753497 | US10383880, Example 82)
Affinity DataEC50:  438nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140702(CHEMBL3753702 | US10383880, Example 3)
Affinity DataEC50:  516nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140703(CHEMBL3754134 | US10383880, Example 2)
Affinity DataEC50:  197nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM56256(MLS000110334 | N-(3-carbazol-9-yl-2-hydroxy-propyl...)
Affinity DataEC50:  870nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140732(CHEMBL3753313)
Affinity DataEC50: >1.00E+4nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140736(CHEMBL3754710 | US10383880, Example 58)
Affinity DataEC50:  308nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140749(CHEMBL3752740 | US10383880, Example 71)
Affinity DataEC50:  532nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140753(CHEMBL3752876)
Affinity DataEC50:  3.53E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140756(CHEMBL3753763)
Affinity DataEC50:  819nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140758(CHEMBL3752125 | US10383880, Example 133)
Affinity DataEC50:  1.27E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140759(CHEMBL3752021 | US10383880, Example 128)
Affinity DataEC50:  690nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140764(CHEMBL3754396)
Affinity DataEC50:  1.02E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140765(CHEMBL1446115 | US10383880, Example 23)
Affinity DataEC50:  272nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140769(CHEMBL3754502)
Affinity DataEC50:  2.55E+3nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140884(CHEMBL3752425)
Affinity DataEC50:  400nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140885(CHEMBL3752453 | US10383880, Example 24)
Affinity DataEC50:  939nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140886(CHEMBL3753460 | US10383880, Example 44)
Affinity DataEC50:  818nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140887(CHEMBL3753709)
Affinity DataEC50:  190nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140888(CHEMBL3753839 | US10383880, Example 20)
Affinity DataEC50:  144nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140889(CHEMBL3752502 | US10383880, Example 33)
Affinity DataEC50:  173nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140890(CHEMBL3754594)
Affinity DataEC50:  73nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140891(CHEMBL3753487)
Affinity DataEC50:  42nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140892(CHEMBL3752737)
Affinity DataEC50:  132nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM50140893(CHEMBL3753932 | US10383880, Example 123)
Affinity DataEC50:  384nMAssay Description:Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythmsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356633(1-(3-(9H-carbazol-9-yl)-2-hydroxypropyl)piperidin-...)
Affinity DataEC50:  171nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356634(1-(3-(9H-carbazol- 9-yl)-2- hydroxypropyl)-3- fluo...)
Affinity DataEC50:  61nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356635(1-(3-(9H-carbazol- 9-yl)-2- hydroxypropyl)-3- meth...)
Affinity DataEC50:  736nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356636(US10214507, Compound 71 | US10759777, Compound 71)
Affinity DataEC50:  188nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356638(1-(3-(9H-carbazol- 9-yl)-2- hydroxypropyl) tetrahy...)
Affinity DataEC50:  299nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356639(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  389nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356640(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  192nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356641(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  1.11E+3nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeriod circadian protein homolog 2(Homo sapiens (Human))
Reset Therapeutics

Curated by ChEMBL
LigandPNGBDBM356642(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxy-2...)
Affinity DataEC50:  536nMAssay Description:Compounds were screened by using a high-throughput circadian assay system as previously described in Zhang, E. E. et al. Cell, 2009, 139, 199-210. In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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