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Found 4 Enz. Inhib. hit(s) with Target = 'Polypeptide N-acetylgalactosaminyltransferase 1'
TargetPolypeptide N-acetylgalactosaminyltransferase 10(Homo sapiens)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50:  330nMAssay Description:Inhibition of catalytic activity of ppGalNAcT10 (unknown origin) using EA2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolypeptide N-acetylgalactosaminyltransferase 14(Homo sapiens)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50:  460nMAssay Description:Inhibition of catalytic activity of ppGalNAcT14 (unknown origin) using EA2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolypeptide N-acetylgalactosaminyltransferase 1(Homo sapiens)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibition of catalytic activity of ppGalNAcT1 (unknown origin) using EA2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolypeptide N-acetylgalactosaminyltransferase 13(Homo sapiens)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of catalytic activity of ppGalNAcT13 (unknown origin) using EA2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed