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Found 23 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha/beta/gamma type'
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  2.70nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136008(12-(3-hydroxypropyl)-9-isopropoxymethyl-6,7,12,13-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50009723(2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229926(CHEMBL319584)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229931(CHEMBL100713)
Affinity DataIC50:  3.40E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229930(CHEMBL97997)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229920(CHEMBL101142)
Affinity DataIC50:  3.60E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229928(CHEMBL97998)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229921(CHEMBL99372)
Affinity DataIC50:  4.50E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229917(CHEMBL100289)
Affinity DataIC50:  4.50E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229932(CHEMBL97921)
Affinity DataIC50:  4.60E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229922(CHEMBL98968)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of [3H]-phorbol dibutyrate binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229924(CHEMBL99156)
Affinity DataIC50:  5.10E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229929(CHEMBL98337)
Affinity DataIC50:  5.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  5.70E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229927(CHEMBL319666)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229916(CHEMBL322371)
Affinity DataIC50:  7.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229933(CHEMBL98542)
Affinity DataIC50:  7.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229915(CHEMBL101358)
Affinity DataIC50:  9.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229925(CHEMBL433408)
Affinity DataIC50:  1.02E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229923(CHEMBL317827)
Affinity DataIC50:  1.54E+5nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229919(CHEMBL101538)
Affinity DataIC50:  1.59E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229918(CHEMBL101731)
Affinity DataIC50:  2.99E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed