Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with Target = 'Sarcoplasmic/endoplasmic reticulum calcium ATPase 2'
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527071(CHEMBL4514624)
Affinity DataKi:  1.30nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50453611(CHEMBL4207081)
Affinity DataKi:  11nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50453612(CHEMBL4216774)
Affinity DataKi:  27nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527068(CHEBI:17734 | CHEMBL468766)
Affinity DataIC50:  90nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527063(CHEMBL4534285)
Affinity DataIC50:  210nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mus musculus)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50410532(4-NONYLPHENOL)
Affinity DataIC50:  350nMAssay Description:Inhibition of SERCA2b in mouse testicular microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM176764(2,5-Di-tert-butylhydroquinone | CAS# 88-58-4 | US9...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rattus norvegicus)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM29608(Bisphenol A (BPA) | Diphenylolpropane | US9688816,...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat cerebellar microsomes SERCA2b by enzyme-coupled methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50854(MLS000028812 | PAXILLINE | SMR000058863 | cid_1050...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rattus norvegicus)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)
Affinity DataIC50:  6.72E+3nMAssay Description:Inhibition of Wistar rat heart SERCA2a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Homo sapiens)
University Of Chemistry And Technology Prague

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed