Found 20 Enz. Inhib. hit(s) with Target = 'Solute carrier family 2, facilitated glucose transporter member 4'
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Antagonist activity at GLUT4 in rat adipocytes assessed as reduction in insulin-stimulated [3H]2-deoxyglucose uptake preincubated for 1 min followed ...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at rat C-terminal 6His/Myc-tagged GLUT4 assessed as reduction in 2-[3H]deoxyglucose uptake measured after 6 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.82E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Homo sapiens)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.52E+5nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 47nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 650nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Rattus norvegicus)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair