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Found 6 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 5'
TargetSolute carrier family 22 member 5(Rattus norvegicus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50375327(CHEMBL410874)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of rat kidney brush border membrane OCTN2 transporter assessed as [3H]carnitine uptake after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Rattus norvegicus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50375326(CHEMBL260616)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of rat kidney brush border membrane OCTN2 transporter assessed as [3H]carnitine uptake after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50103624(40602 | CHEBI:3537 | Cefaloridine | Cephaloridine ...)
Affinity DataIC50:  2.30E+5nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Rattus norvegicus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50375328(CHEMBL410276)
Affinity DataIC50:  4.43E+5nMAssay Description:Inhibition of rat kidney brush border membrane OCTN2 transporter assessed as [3H]carnitine uptake after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50350470(CEFEPIME | Maxipime)
Affinity DataIC50:  1.70E+6nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50485614(Cefoselis)
Affinity DataIC50:  6.40E+7nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed