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Found 6 Enz. Inhib. hit(s) with Target = 'TAR DNA-binding protein 43'
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544711(CHEMBL4647070)
Affinity DataIC50: <100nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544712(CHEMBL4635203)
Affinity DataIC50:  100nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM67690(1,4-bis[2-(2-hydroxyethylamino)ethylamino]-5,8-bis...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM16435(5-(1,2-dithiolan-3-yl)pentanamide | 5-(dithiolan-3...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50106731((+)-alpha-Lipoic acid | (R)-(+)-lipoic acid | (R)-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTAR DNA-binding protein 43(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544713(CHEMBL4638490)
Affinity DataKd:  8.90E+4nMAssay Description:Binding affinity to TDP-43 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed