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Found 116 Enz. Inhib. hit(s) with Target = 'Telomeric repeat-binding factor 2'
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136318(CHEMBL3752561)
Affinity DataKi:  7nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136317(CHEMBL3752190)
Affinity DataKi:  16nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136319(CHEMBL3752814)
Affinity DataKi:  19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136315(CHEMBL3751889)
Affinity DataKi:  19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136320(CHEMBL3752958)
Affinity DataKi:  22nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136311(CHEMBL3752264)
Affinity DataKi:  32nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136310(CHEMBL3754578)
Affinity DataKi:  53nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338579(CHEMBL4166000)
Affinity DataKi:  90nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338579(CHEMBL4166000)
Affinity DataKi:  90nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136316(CHEMBL3752170)
Affinity DataKi:  130nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136305(CHEMBL3752828)
Affinity DataKi:  140nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338573(CHEMBL4163499)
Affinity DataKi:  210nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338561(CHEMBL4172926)
Affinity DataKi:  240nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546773(CHEMBL4782698)
Affinity DataKi:  330nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338565(CHEMBL4176290)
Affinity DataKi:  340nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338580(CHEMBL4163072)
Affinity DataKi:  380nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338572(CHEMBL4161391)
Affinity DataKi:  510nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338555(CHEMBL4161856)
Affinity DataKi:  720nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338574(CHEMBL4159482)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136300(CHEMBL3752803)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136313(CHEMBL3752883)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338567(CHEMBL4160402)
Affinity DataKi:  1.89E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136314(CHEMBL3752069)
Affinity DataKi:  2.00E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136309(CHEMBL3754122)
Affinity DataKi:  2.10E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338564(CHEMBL4168423)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136301(CHEMBL3753586)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338583(CHEMBL4167227)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338558(CHEMBL4169779)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546766(CHEMBL4745325)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546787(CHEMBL4792503)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338570(CHEMBL4168052)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546783(CHEMBL4759024)
Affinity DataKi:  4.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546775(CHEMBL4746160)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546776(CHEMBL4750127)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136312(CHEMBL3753717)
Affinity DataKi:  5.80E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338581(CHEMBL4166947)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136305(CHEMBL3752828)
Affinity DataKi:  6.20E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546782(CHEMBL4745167)
Affinity DataKi:  6.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338556(CHEMBL4165033)
Affinity DataKi:  8.50E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546774(CHEMBL4779157)
Affinity DataKi:  8.80E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546784(CHEMBL4744656)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338563(CHEMBL4176438)
Affinity DataKi:  1.12E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338560(CHEMBL4174183)
Affinity DataKi:  1.13E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546788(CHEMBL4754108)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546769(CHEMBL4758244)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136306(CHEMBL3754019)
Affinity DataKi:  1.32E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136307(CHEMBL3754707)
Affinity DataKi:  1.37E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50136302(CHEMBL3752348)
Affinity DataKi:  1.39E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338554(CHEMBL4168576)
Affinity DataKi:  1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546789(CHEMBL4755348)
Affinity DataKi:  1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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