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Found 14 Enz. Inhib. hit(s) with Target = 'Thymidine kinase 2, mitochondrial (Predicted)'
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028586(1-(4-Benzyloxy-5-hydroxymethyl-tetrahydro-furan-2-...)
Affinity DataKi:  8.00E+3nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  1.10E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028587(1-(4-Ethylsulfanyl-5-hydroxymethyl-tetrahydro-fura...)
Affinity DataKi:  6.20E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000966(CHEMBL3143491)
Affinity DataKi:  7.20E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028583(1-(4-Hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl...)
Affinity DataKi:  7.70E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028579(1-(4-Hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl...)
Affinity DataKi:  2.50E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367094(DEOXYCYTIDINE | EN300-6477283)
Affinity DataKi:  3.20E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50018445(1-((2R,5S)-5-(hydroxymethyl)-tetrahydrofuran-2-yl)...)
Affinity DataKi:  8.80E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028581(1-(5-Hexylaminomethyl-4-hydroxy-tetrahydro-furan-2...)
Affinity DataKi:  9.60E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000969(CHEMBL3143490)
Affinity DataKi:  1.10E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028576(1-(5-Ethylaminomethyl-4-hydroxy-tetrahydro-furan-2...)
Affinity DataKi:  1.44E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50132294(1-((2R,4S,5S)-4-amino-5-(hydroxymethyl)-tetrahydro...)
Affinity DataKi:  2.60E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50013111(1-((2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl...)
Affinity DataKi:  3.25E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial (Predicted)(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50132297(1-((2R,4S,5R)-5-(aminomethyl)-4-hydroxy-tetrahydro...)
Affinity DataKi:  4.60E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed