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Found 22 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410]'
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012902(CHEMBL3261318 | USRE46024, 1)
Affinity DataEC50:  7.75E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012908(CHEMBL3261334 | USRE46024, 22)
Affinity DataEC50:  136nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012912(CHEMBL3261321 | USRE46024, 3)
Affinity DataEC50:  519nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012901(CHEMBL3261320 | USRE46024, 4)
Affinity DataEC50:  2.33E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012916(CHEMBL3261322 | USRE46024, 5)
Affinity DataEC50:  699nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012918(CHEMBL3261324 | USRE46024, 6)
Affinity DataEC50:  666nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM60964(USRE46024, 7)
Affinity DataEC50:  117nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012905(CHEMBL3261331 | USRE46024, 8)
Affinity DataEC50:  192nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012915(CHEMBL3261335 | USRE46024, 9)
Affinity DataEC50:  115nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012906(CHEMBL3261323 | USRE46024, 10)
Affinity DataEC50:  767nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM237173(USRE46024, 11)
Affinity DataEC50:  1.20E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012911(CHEMBL3261332 | USRE46024, 12)
Affinity DataEC50:  133nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012907(CHEMBL3261336 | USRE46024, 13)
Affinity DataEC50:  92nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012910(CHEMBL3261326 | USRE46024, 14)
Affinity DataEC50:  2.99E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012917(CHEMBL3261327 | USRE46024, 15)
Affinity DataEC50:  601nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012913(CHEMBL3261333 | USRE46024, 16)
Affinity DataEC50:  66nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012903(CHEMBL3261328 | USRE46024, 17)
Affinity DataEC50:  2.04E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM237174(USRE46024, 18)
Affinity DataEC50:  9.18E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012817(CHEMBL3261330 | USRE46024, 19)
Affinity DataEC50:  6.98E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM237175(USRE46024, 20)
Affinity DataEC50:  7.04E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM237176(USRE46024, 21)
Affinity DataEC50:  3.21E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410](Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50012859(CHEMBL3261319 | USRE46024, 2)
Affinity DataEC50:  7.31E+3nMpH: 7.0Assay Description:Thirty microliters of H6-TRβ (50 nM) in 50 mM Hepes, pH 7.0, 1 mM DTT, 0.05% NP40 and 0.2 mg/ml BSA (Binding Buffer) was mixed with an equal vol...More data for this Ligand-Target Pair
In DepthDetails US Patent