Compile Data Set for Download or QSAR
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Found 11 of ki for UniProtKB: A0A0G4Q818
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24969([(2-{[(benzyloxy)carbonyl]amino}acetamido)methyl](...)
Affinity DataKi:  450nM ΔG°:  -8.80kcal/mole IC50:  3.10E+3nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24971(({[(benzyloxy)carbonyl]amino}methyl)(methyl)sulfan...)
Affinity DataKi:  1.40E+4nM ΔG°:  -6.73kcal/mole IC50:  1.58E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24967(methyl[(methylamino)methyl]phosphinic acid | organ...)
Affinity DataKi:  2.70E+4nM ΔG°:  -6.33kcal/mole IC50:  1.53E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24962([(2-aminoacetamido)methyl](methyl)phosphinic acid ...)
Affinity DataKi:  3.00E+4nM ΔG°:  -6.27kcal/mole IC50:  8.60E+4nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24965(organophosphorus derivative, 6 | {[(2S)-2-amino-3-...)
Affinity DataKi:  3.26E+4nM ΔG°:  -6.22kcal/mole IC50:  1.83E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24966(organophosphorus derivative, 7 | {[(2S)-2-amino-3-...)
Affinity DataKi:  4.10E+4nM ΔG°:  -6.08kcal/mole IC50:  3.42E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24968(({[(benzyloxy)carbonyl]amino}methyl)(methyl)phosph...)
Affinity DataKi:  6.50E+4nM ΔG°:  -5.80kcal/mole IC50:  3.19E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24964(organophosphorus derivative, 5 | {[(2S)-2-amino-3-...)
Affinity DataKi:  1.76E+5nM ΔG°:  -5.20kcal/mole IC50:  7.54E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24970([(2-{[(benzyloxy)carbonyl]amino}acetamido)methyl](...)
Affinity DataKi:  1.78E+5nM ΔG°:  -5.20kcal/mole IC50:  6.40E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24963(organophosphorus derivative, 4 | {[(2S)-2-amino-3-...)
Affinity DataKi:  2.08E+5nM ΔG°:  -5.10kcal/mole IC50:  6.17E+5nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24960((aminomethyl)(methyl)phosphinic acid | organophosp...)
Affinity DataKi:  4.25E+5nM ΔG°:  -4.67kcal/mole IC50:  2.53E+6nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed