Affinity DataIC50: 2nMAssay Description:Binding affinity against human estrogen receptor beta (ER beta) in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity against human estrogen receptor alpha in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18.6nMAssay Description:The binding affinity and selectivity of candidate molecules yielded from
database screening were determined by a fluorescent polarization
competiti...More data for this Ligand-Target Pair
Affinity DataIC50: 18.6nMAssay Description:Binding affinity for human Estrogen receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 18.6nMAssay Description:Binding affinity for human Estrogen receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 75.7nMAssay Description:Binding affinity for human Estrogen receptor AlphaMore data for this Ligand-Target Pair
Affinity DataIC50: 75.7nMAssay Description:Binding affinity for human Estrogen receptor AlphaMore data for this Ligand-Target Pair
Affinity DataIC50: 75.7nMAssay Description:The binding affinity and selectivity of candidate molecules yielded from
database screening were determined by a fluorescent polarization
competiti...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
University Of Padua And Institute Of Biomolecular Chemistry
Curated by ChEMBL
University Of Padua And Institute Of Biomolecular Chemistry
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human CK2 using HRRRDDD-SDDD-NH2 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at human PXR transfected in African green monkey CV1 cells assessed as inhibition of SR12813-induced transactivation after 24 hrs...More data for this Ligand-Target Pair
Affinity DataIC50: >4.27E+4nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair