TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of ovine COX1 after 5 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant COX2 after 5 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Zafes/Liff/Goethe University Frankfurt
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of gamma-secretase in HEK293 cells co-overexpressing NotchdeltaE assessed as inhibition of notch cleavage by luciferase reporter gene assa...More data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.71E+4nMAssay Description:Displacement of [3H]L685458 from gamma-secretase in human THP1 cellsMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.25E+4nMAssay Description:Inhibition of gamma-secretase in HEK293 cells co-overexpressing APP Swedish mutant assessed as inhibition of amyloid beta 42 production by luciferase...More data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.15E+5nMAssay Description:Inhibition of gamma-secretase in HEK293 cells co-overexpressing APP Swedish mutant assessed as inhibition of amyloid beta 40 production by luciferase...More data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.32E+5nMAssay Description:Displacement of [3H]IN973 from gamma-secretase in human THP1 cellsMore data for this Ligand-Target Pair