Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 81467
TargetSerine protease hepsin(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center

US Patent
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50:  2.02E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
Fred Hutchinson Cancer Research Center

US Patent
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50: >2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProthrombin(Bos taurus (Bovine))
Fred Hutchinson Cancer Research Center

US Patent
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50: >2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCruzipain(Trypanosoma cruzi)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine preincubated for 5 mins before substrate addition by fluorescence assay in absence of Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine preincubated for 5 mins before substrate addition by fluorescence assay in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed