Affinity DataKd: 0.0360nMAssay Description:Binding constant for JAK2(JH1domain-catalytic) kinase domainMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 0.900nMAssay Description:Binding constant for TYK2(JH1domain-catalytic) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding constant for JAK3(JH1domain-catalytic) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.40nMAssay Description:Binding constant for JAK1(JH1domain-catalytic) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Binding affinity to human recombinant N-terminal hexahistidine tagged JAK2 JH1 catalytic domain (835 to 1132 residues) expressed in baculovirus infec...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 41nMAssay Description:Binding constant for MAP3K2 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 46nMAssay Description:Binding constant for CAMK2A kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Binding constant for ROCK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 68nMAssay Description:Binding constant for DCAMKL1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding constant for DAPK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 89nMAssay Description:Binding constant for DAPK3 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit delta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 90nMAssay Description:Binding constant for CAMK2D kinase domainMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 90nMAssay Description:Binding constant for LRRK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Binding constant for GAK kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 120nMAssay Description:Binding constant for CAMK1D kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding constant for AAK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding constant for RSK1(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding constant for PLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for RPS6KA5(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for RSK3(Kin.Dom.1-N-terminal) kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for MAP3K3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for RSK4(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for ULK2 kinase domainMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding constant for RET(V804M) kinase domainMore data for this Ligand-Target Pair
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding constant for MKNK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for PLK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding constant for DCAMKL3 kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 19(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 270nMAssay Description:Binding constant for YSK4 kinase domainMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 280nMAssay Description:Binding constant for RET(V804L) kinase domainMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding constant for LRRK2 kinase domainMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding constant for IRAK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding constant for ULK1 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 310nMAssay Description:Binding constant for CAMK2B kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding constant for TAOK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding constant for SNARK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 340nMAssay Description:Binding constant for RPS6KA4(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 360nMAssay Description:Binding constant for MYLK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Binding constant for TRKB kinase domainMore data for this Ligand-Target Pair
TargetAnkyrin repeat and protein kinase domain-containing protein 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 390nMAssay Description:Binding constant for ANKK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding constant for LTK kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Comenius University In Bratislava
Curated by ChEMBL
Comenius University In Bratislava
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding affinity to recombinant human CLK2 (D144 to R498 residues) expressed in bacterial expression system by KinomeScan assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Comenius University In Bratislava
Curated by ChEMBL
Comenius University In Bratislava
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding constant for MEK3 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding constant for CAMK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 480nMAssay Description:Binding constant for TTK kinase domainMore data for this Ligand-Target Pair