Compile Data Set for Download or QSAR
maximum 50k data
Found 27 of ki for monomerid = 214799
TargetKappa-type opioid receptor [D138N](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [M142A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  20nM ΔG°:  -43.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [D138A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  30nM ΔG°:  -42.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [K227A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  51nM ΔG°:  -41.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [H291F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  65nM ΔG°:  -41.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [K212A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  100nM ΔG°:  -40.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [E297A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  110nM ΔG°:  -39.7kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [M226A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  180nM ΔG°:  -38.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [K200A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  180nM ΔG°:  -38.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [I135A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  220nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  220nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y139F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  300nM ΔG°:  -37.2kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y312F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  340nM ΔG°:  -36.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y139A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  350nM ΔG°:  -36.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y312A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  390nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [H291A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  390nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y320F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  470nM ΔG°:  -36.1kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [I294A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  480nM ΔG°:  -36.1kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y313F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  510nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y119F](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  520nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y66A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  550nM ΔG°:  -35.7kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Q115A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  580nM ΔG°:  -35.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [I316A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  890nM ΔG°:  -34.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  1.30E+3nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y313A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  2.20E+3nM ΔG°:  -32.3kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y320A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  4.20E+3nM ΔG°:  -30.7kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor [Y119A](Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM214799(1xx)
Affinity DataKi:  5.50E+3nM ΔG°:  -30.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed as previously detailed [Yan et al., Biochemistry, 48:6898-6908]. In brief, crude cell membranes were prepar...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed