TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat Sprague-Dawley kidney membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
Affinity DataKi: 7.30nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 23nM ΔG°: -40.5kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membranes by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]PK11195 from translocator protein in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to peripheral benzodiazepine receptors using [3H]-PK11195 radioligand in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of [3H]PK11195 binding to TSPO in rat kidney mitochondrial membranesMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
Affinity DataKi: 34nMAssay Description:Displacement of [3H]PK11195 from PBR in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
Technion-Israel Institute Of Technology
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Tokyo Dental College
Curated by PDSP Ki Database
Tokyo Dental College
Curated by PDSP Ki Database