Affinity DataKi: 16nMAssay Description:Inhibitory constant against calcium channel receptors (CCRs)More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of CYP3A4-mediated N-demethylation in human liver microsomesMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Johns Hopkins University
Curated by PDSP Ki Database
Johns Hopkins University
Curated by PDSP Ki Database
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Johns Hopkins University
Curated by PDSP Ki Database
Johns Hopkins University
Curated by PDSP Ki Database
Affinity DataKi: 280nMAssay Description:Calcium antagonistic activity by measuring [3H]-nitrendipine displacement from rat heart L-type [Ca2+] channelMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Johns Hopkins University
Curated by PDSP Ki Database
Johns Hopkins University
Curated by PDSP Ki Database
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:Displacement of [3H]-diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Mechanism based inhibition of human cytochrome P450 3A4 measured by testosterone 6-beta hydroxylationMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Mechanism based inhibition of human cytochrome P450 3A4 measured by midazolam hydroxylase activityMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Johns Hopkins University
Curated by PDSP Ki Database
Johns Hopkins University
Curated by PDSP Ki Database
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Johns Hopkins University
Curated by PDSP Ki Database
Johns Hopkins University
Curated by PDSP Ki Database