TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataKi: 460nM ΔG°: -36.2kJ/molepH: 7.0 T: 2°CAssay Description:Assays were conducted at 25 C in 20 mM sodium phosphate buffer (pH 7.0) and 0.01% bovine serum albumin unless otherwise noted. AChE concentrations we...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Bath
Curated by PDSP Ki Database
University Of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Bath
Curated by PDSP Ki Database
University Of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Bath
Curated by PDSP Ki Database
University Of Bath
Curated by PDSP Ki Database
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity to mouse AChEMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Kentucky
Curated by ChEMBL
University Of Kentucky
Curated by ChEMBL
Affinity DataKi: 5.73E+3nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha4-beta2 was evaluated by its ability to inhibit [3H]NIC binding to rat brain membranesMore data for this Ligand-Target Pair
TargetCholinergic receptor nicotinic alpha 6 subunit(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Chick)
University Of Milan
Curated by PDSP Ki Database
University Of Milan
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Bath
Curated by PDSP Ki Database
University Of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Kentucky
Curated by ChEMBL
University Of Kentucky
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity nicotinic acetylcholine receptor alpha-7 was evaluated by its ability to inhibit [3H]methyllycaconitine ([3H]-MLA) binding to rat br...More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+6nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair