TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to salt water mollusc Aplysia californica AChBP Y55W mutant assessed as [3H]acetamiprid binding by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Potency to displace [3H]-Nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 immuno-isolated from M10 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 970nMAssay Description:Binding affinity to freshwater snail Lymnaea stagnalis AChBP assessed as [3H]EPI binding by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AF-DX 384 from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]QNB from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair