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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50403163'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50403163(OXITRIPTAN)
Affinity DataEC50:  130nMAssay Description:Agonist activity at 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding incubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50403163(OXITRIPTAN)
Affinity DataEC50:  1.35nMAssay Description:Agonist activity at recombinant human 5HT2A receptor expressed in Flp-In-293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50403163(OXITRIPTAN)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at recombinant human 5HT2A receptor expressed in Flp-In-293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed