Found 28 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM21398'
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Affinity DataKi: 2.51E+3nMAssay Description:In vitro ability to displace [3H]mesulergine binding from 5-hydroxytryptamine 2C receptor from bovine choroid plexus.More data for this Ligand-Target Pair
Affinity DataKi: 3.95E+3nMAssay Description:Binding assay using 5-HT2A, Dopamine D2, SERT, αA1, 5-HT2C and H1 Receptors.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of [3H]Mesulergine from rat 5-HT2C receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Binding affinity to human cloned 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity towards human serotonin 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.24E+3nMAssay Description:Displacement of [3H]mesulergine human cloned serotonin 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.24E+3nMAssay Description:Binding affinity towards serotonin 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.24E+3nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.24E+3nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [3H]-mesulergine binding to 5-hydroxytryptamine 2C receptor in rat brain membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck
Curated by PDSP Ki Database
H. Lundbeck
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity towards 5-hydroxytryptamine 2C receptor in membranes from pig choroid plexus using [3H]-N-methyl-mesulergineMore data for this Ligand-Target Pair