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Found 4 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50169601'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50169601(1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylm...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50169601(1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylm...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity against h5-HT6 receptor transiently expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50169601(1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylm...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-LSD from cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50169601(1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylm...)
Affinity DataIC50:  81.4nMAssay Description:Inhibition of cAMP production in HeLa cells expressing human 5-HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed