Found 16 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 7' and Ligand = 'BDBM50001885'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-5-CT from human 5-HT7R expressed in HEK293 cell membranes after 1 hr at 37 degC by microbeta counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataKi: 1.40nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-5-CT from 5-HT7 receptor in rat hypothalamus homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibition of [3H]-5-HT binding to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataKi: 12.8nMAssay Description:5-HT7: (1) The prepared membrane was applied with buffer, and homogenizer was used for evenly dispersing. 15 tubes were mixed into a 100 ml container...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataKi: 41nMAssay Description:Displacement of [3H]5-CT from rat cerebral cortex 5HT7 receptor measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair