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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50037971'
TargetAdenosine receptor A1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50037971(CHEMBL3359414)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50037971(CHEMBL3359414)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at human recombinant adenosine A1 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed